BDBM50399620 CHEMBL2181187

SMILES CCCN1CCC(COc2nc3c(OC)cccc3c3ccccc23)CC1

InChI Key InChIKey=OLINRUQQUFMPJJ-UHFFFAOYSA-N

Data  13 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50399620   

Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399620(CHEMBL2181187)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]GR113808 from human recombinant 5HT4R expressed in HEK293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50399620(CHEMBL2181187)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399620(CHEMBL2181187)
Affinity DataEC50:  79.4nMAssay Description:Inverse agonist activity at human recombinant 5HT4R expressed in HEK293T cells assessed as Gs activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed